Intermediates for Anticoagulant
| APPLICATION | PRODUCTS CAS No. |
|---|---|
| Apixaban | |
| Clopidogrel |
5402-55-1 30433-91-1 4,5,6,7-Tetrahydrothieno[3,2,c] pyridine HCl 28783-41-7 |
| Edoxaban | |
| Rivaroxaban |
5-Chlorothiophene-2-carboxylic acid 24065-33-6 (S)-(+)-N-(2,3-epoxypropyl)phthalimide 161596-47-0 4-(4-Aminophenyl)morpholin-3-one 438056-69-0 |
| Ticagrelor |
4,6-Dichloro-2-propylthiopyrimidine-5-amine 145783-15-9 (1R,2S)-2-(3,4-difluorophenyl)cyclopropanamine HCl 1156491-10-9 |
Intermediates for Antihypertensive
Intermediates for Weight-loss
Intermediates for Antimicrobial
| APPLICATION | PRODUCTS CAS No. |
|---|---|
| Biapenem |
153851-71-9 |
| Doripenem |
491878-06-9 |
| Ertapenem | |
| Imipenem |
P-nitrobenzyl-6-(1-hydroxyethyl)-1-azabicyclo(3.2.0)-heptane-3,7-dione-2-carboxylate (BCK) 74288-40-7 90776-58-2 |
| Isavuconazole |
20099-89-2 2-(Methylamino)pyridine-3-methanol 32399-12-5 |
| Meropenem |
96034-64-9 Meropenem trihydrate non sterile 96036-03-2 |
| Posaconazole |
[(2S,3S)-2-(benzyloxy)pentan-3-yl]hydrazine 183871-36-5 |
| Tebipenem |
179337-57-6 |
| Other KSM |
Tert-butyl dimethyl silyl chloride (TBDMS) 18162-48-6 Beta-methyl vinyl phosphate (MAP) 90776-59-3 |
Intermediates for CNS agents
| APPLICATION | PRODUCTS CAS No. |
|---|---|
| Atogepant | |
| Duloxetine |
321-38-0 |
| Paroxetine | |
| Rimegepant |
1190363-46-2 1289024-42-5 |
| Suzetrigine |
(R)-4,4,4-trifluoro-3-hydroxy-3-methylbutan-2-one 2875067-31-3 Methyl 4-aminopyridine-2-carboxylate 71469-93-7 |
| Ubrogepant |
Intermediates for Antiviral
| APPLICATION | PRODUCTS CAS No. |
|---|---|
| Baloxavir marboxil |
7,8-Difluoro-6,11-dihydrodibenzo[b,e]thiepin-11-ol 1985607-83-7 2136287-62-0 2136287-61-9 |
| Bictegravir |
(1R,3S)-3-aminocyclopentanol HCl 1279032-31-3 |
| Glecaprevir | |
| Pibrentasvir | |
| Voxilaprevir |
1799733-54-2 |
Intermediates for Anticancer
| APPLICATION | PRODUCTS CAS No. |
|---|---|
| Bortezomib |
(R)-boroleu-(+)-pinanediol trifluoroacetate 179324-87-9 |
| Docetaxel |
90332-66-4 90332-63-1 10-Deacetyl baccatin III(10-DAB) 32981-86-5 |
| Encorafenib |
1269440-69-8 |
| Gedatolisib |
4-(4,6-Dimorpholino-1,3,5-triazin-2-yl)aniline 1197159-91-3 23138-53-6 |
| Infigratinib |
4-(4-Ethylpiperazin-1-ly)aniline 115619-01-7 4-Chloro-6-methylaminopyrimidine 65766-32-7 2,6-Dichloro-3,5-dimethoxybenzenamine 872509-56-3 |
| Ivosidenib |
10386-27-3 210169-05-4 3-Oxocyclobutanecarboxylic acid 23761-23-1 3,3-Difluorocyclobutanamine HCl 637031-93-7 |
| Niraparib |
3-Formyl-2-nitrobenzoic acid methyl ester 138229-59-1 |
| Olaparib |
218301-22-5 |
| Palbociclib | |
| Ribociclib | |
| Ruxolitinib |
(betaR)-beta-cyclopentyl-4-(7H-pyrrolo[2,3-d] pyrimidin-4-yl)-1H-pyrazole-1-propanenitrile phosphate 1092939-17-7 1146629-84-6 3-Cyclopentyl-3-[4-(4,4,5,5-tetramethyl-1,3,2- dioxaborolan-2-yl)-1H-pyrazol-1-yl]propanenitrile 1153949-38-2 1187595-88-5 |
| Trametinib |
516-05-2 |
| Zanubrutinib |
Intermediates for Anti-Diabetic
| APPLICATION | PRODUCTS CAS No. |
|---|---|
| Dapagliflozin |
90-80-2 4-(5-Bromo-2-chlorobenzyl)phenyl ethyl ether 461432-23-5 461432-25-7 |
| Empagliflozin |
(S)-(+)-3-hydroxytetrahydrofuran 86087-23-2 915095-99-7 |
| Ertugliflozin |
1528636-39-6 |
| Linagliptin |
1076-22-8 3355-28-0 93703-24-3 8-Bromo-7-(2-butyn-1-yl)-3-methylxanthine 666816-98-4 309956-78-3 (R)-3-Piperidinamine dihydrochloride 334618-23-4 |
| Saxagliptin |
Boc-3-hydroxy-1-adamantyl-D-glycine 361442-00-4 |
| Sitagliptin | |
| Vildagliptin |
281-23-2 702-82-9 665-66-7 |
Intermediates for Lipid-lowering
| APPLICATION | PRODUCTS CAS No. |
|---|---|
| Atorvastatin |
Ethyl (R)-(-)-4-cyano-3-hydroxybutyrate (A5) 141942-85-0 |
| Enlicitide |
Fmoc-3-(boc-aminomethyl)-Phe-OH 266999-24-0 3067192-76-8 167275-47-0 103336-06-7 188970-92-5 77128-72-4 |
| Rosuvatatin |
4-(4-Fluorophenyl)-6-isopropyl-2-[(N-methyl-n- methylsulfonyl)amino]pyrimidine-5-yl-methanol (Z7) 147118-36-3 |
Intermediates for Antimalarial
| APPLICATION | PRODUCTS CAS No. |
|---|---|
| Artemether |
63968-64-9 |
| Atovaquone |
130-15-4 |
| Lumefantrine |
86-73-7 104-88-1 7012-16-0 2-(2,7-Dichloro-9H-fluoren-4-yl)oxirane 53221-14-0 |
| Sulphadoxine |
63-74-1 95-92-1 6290-49-9 4,6-Dichloro-5-methoxypyrimidine 5018-38-2 |
Intermediates for Other Categories
| APPLICATION | PRODUCTS CAS No. |
|---|---|
| Carbamazepine / Oxcarbazepine |
494-19-9 Iminodibenzyl carbonyl chloride(IDBCC) 33948-19-5 Iminostilbene carbonyl chloride(ISBCC) 33948-22-0 10-Methoxyiminostilbene(10-MISB) 4698-11-7 |
| Elinzanetant | |
| Eltrombopag | |
| Etodolac |
30414-53-0 41340-36-7 200880-31-5 |
| Etrasimod | |
| Febuxostat | |
| Finerenone |
65193-87-5 21962-45-8 4-Amino-5-methyl-2(1H)-pyridinone 95306-64-2 2640574-73-6 |
| Iguratimod | |
| Iptacopan |
Methyl 4-[(2S,4S)-4-ethoxy-2-piperidyl]benzoate 1644667-61-7 |
| Mirogabalin |
3-Ethylbicyclo[3.2.0]hept-3-en-6-one 1235479-59-0 (1R,5S)-3-ethyl-bicyclo[3.2.0]hept-3-en-6-one 1235479-61-4 |
| Silodosin | |
| Tofacitinib |
4-Chloro-7H-pyrrolo[2,3-d]pyrimidine 3680-69-1 2,4-Dichloro-7H-pyrrolo[2,3-d]pyrimidine 90213-66-4 Benzyl-N,4-dimethylpiperidin-3-amine dihydrochloride 1228879-37-5 3-Bis(4-methylbenzoyloxy)succinate) 477600-71-8 |
| Upadacitinib |
875781-43-4 1708997-42-5 |
| Vonoprazan |
16133-25-8 5-(2-Fluorophenyl)-1H-pyrrole-3-carbaldehyde 881674-56-2 |
| Vibegron |

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